Products for Research Use Only

TP003

CAT: 0931-T23466-01Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0931-T23466-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
628690-75-5
Target
GABA Receptor
Related Pathways
Neuroscience, Membrane transporter/Ion channel
Purity
0.9917
Bioactivity
TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.64 nM, respectively. TP003 has antianxiety and partial anticonvulsant activity via the α2GABAA receptor.
Smiles
FC=1C=2N(C(=CN2)C3=CC(=C(F)C=C3)C4=C(C#N)C=C(F)C=C4)C=CC1C(C)(C)O
Molecular Formula
C23H16F3N3O
Molecular Weight
407.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
532821TP003