KDM2/7-IN-1

• Target:

  Histone Demethylase

• Related Pathways:

  Chromatin/Epigenetic

• Purity:

  0.9987

• Bioactivity:

  KDM2/7-IN-1 (TC-E 5002) is a selective small-molecule inhibitor of the KDM2/7 histone demethylase subfamily, exhibiting IC50 values of 0.2, 1.2, 6.8, 55, 83, >100, and >120 ?M for KDM7A, KDM7B, KDM2A, KDM5A, KDM4C, KDM6A, and KDM4A, respectively. KDM2/7-IN-1 inhibits the proliferation of HeLa and KYSE-150 cancer cells in vitro, highlighting its utility in epigenetic and oncology research.

• Smiles:

  O=C (O) CCN (O) C (=O) CCCCCCCCC1CC1

• Molecular Formula:

  C15H27NO4

• Molecular Weight:

  285.38

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1453071-47-0