Proxyfan

• CAS Number :

  177708-09-7

• Target :

  Histamine Receptor

• Related Pathways :

  Neuroscience|||Immunology/Inflammation|||GPCR/G Protein

• Purity :

  0.9968

• Bioactivity :

  Proxyfan (Proxifan) is a high-affinity protean antagonist/agonist of histamine H3 receptors with a full spectrum of pharmacological activity ranging from full agonist to full inverse agonist (antagonist), depending on the competition between constitutively active and resting H3 receptors within a given tissue or brain region.Proxyfan acts as a neutral antagonist in the feeding-associated ventral medial nucleus of the hypothalamus, and as a agonist in the basolateral amygdala of the rat (BLA) .

• Smiles :

  N1=CNC(=C1)CCCOCC=2C=CC=CC2

• Molecular Formula :

  C13H16N2O

• Molecular Weight :

  216.28

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C