L-365260

• Target :

  Cholecystokinin Receptor

• Related Pathways :

  GPCR/G Protein

• Purity :

  0.9975

• Bioactivity :

  L-365260 is an orally available, selective and potent nonpeptide gastrin and cerebral cholecystokinin receptor (CCK-B) antagonist.L-365260 inhibits CCK-8S-induced increase in [Ca2+]i, blocks stress-induced hypersensitivity in viscera, and blocks the anti-exploratory effect of CCK-4.L-365260 has been used in the study of neurological Ojibwa and endocrine diseases.

• Smiles :

  CN1c2ccccc2C(=N[C@@H](NC(=O)Nc2cccc(C)c2)C1=O)c1ccccc1

• Molecular Formula :

  C24H22N4O2

• Molecular Weight :

  398.46

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  118101-09-0