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INCB054329

CAT: 0931-T22345-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T22345-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1628607-64-6
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.9952
Bioactivity
INCB054329, a structurally distinct bromodomain and extraterminal domain (BET) inhibitor, inhibits BRD2-BD1, BRD2-BD2, BRD3-BD1, BRD3-BD2, BRD4-BD1, BRD4-BD2, BRDT-BD1 and BRDT-BD2 with IC50 values of 44 nM, 5 nM, 9 nM, 1 nM, 28 nM, 3 nM, 119 nM and 63 nM respectively.
Smiles
Cc1noc(C)c1-c1ccc2[nH]c(=O)n3[C@H](COc1c23)c1ccccn1
Molecular Formula
C19H16N4O3
Molecular Weight
348.36
Shipping Conditions
Ice Packs
Storage Temperature
-20°C