XAV-939
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


XAV-939
Target:
PARP|||Wnt/beta-cateninRelated Pathways:
Stem Cells|||Chromatin/Epigenetic|||Cytoskeletal Signaling|||DNA Damage/DNA RepairPurity:
0.9967Bioactivity:
XAV-939 (NVP-XAV939) is a Tankyrase (TNKS) inhibitor that inhibits TNKS1 and TNKS2 (IC50=11/4 nM) . XAV-939 selectively inhibits Wnt/?-catenin-mediated transcription.Smiles:
FC(F)(F)C1=CC=C(C=C1)C1=NC(=O)C2=C(CCSC2)N1Molecular Formula:
C14H11F3N2OSMolecular Weight:
312.31Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
284028-89-3
