Products for Research Use Only

TPOP146

CAT: 0931-T17147Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0931-T17147Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2018300-62-2
Target
Epigenetic Reader Domain, Histone Acetyltransferase
Related Pathways
Chromatin/Epigenetic
Bioactivity
TPOP146 is a selective CBP/P300 benzoxazepine bromodomain inhibitor with Kd values of 134 nM for CBP and 5.02 μM for BRD4.
Smiles
CCC(=O)N1CCOc2c(C1)cc(cc2C(=O)N[C@H]1CCCN(C)C1)-c1cc(OC)cc(OC)c1
Molecular Formula
C27H35N3O5
Molecular Weight
481.58
Shipping Conditions
Ice Packs
Storage Temperature
-20°C