Timapiprant sodium

• Target:

  Others|||Prostaglandin Receptor

• Related Pathways:

  GPCR/G Protein|||Immunology/Inflammation|||Others

• Bioactivity:

  Timapiprant sodium inhibits mast cell activation of Th2 lymphocytes and eosinophils. Timapiprant sodium is a potent and selective D prostanoid receptor 2 antagonist. Timapiprant sodium potently displaces [3H] PGD2 from human recombinant DP2 (Ki=13 nM), rat recombinant DP2 (Ki=3 nM), human native DP2 (Ki=4 nM) .

• Smiles:

  [Na].Cc1c(Cc2ccc3ccccc3n2)c2cc(F)ccc2n1CC(O)=O

• Molecular Formula:

  C21H17FN2NaO2

• Molecular Weight:

  371.367

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  950688-14-9