TAK-243

CAT: 0931-T16974-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-T16974-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1450833-55-2
Target
NF-?B|||Apoptosis|||E1/E2/E3 Enzyme
Related Pathways
Apoptosis|||NF-?B|||Ubiquitination
Purity
0.9893
Bioactivity
TAK-243 (MLN7243) is a selective inhibitor of the ubiquitin-activating enzyme UAE (IC50=1 nM), blocking ubiquitin binding and disrupting both mono-ubiquitin signaling and overall protein ubiquitination. TAK-243 exhibits antitumor activity and promotes apoptosis.
Smiles
NS(=O)(=O)OC[C@H]1C[C@@H](Nc2ccnc3cc(nn23)-c2cccc(SC(F)(F)F)c2)[C@H](O)[C@@H]1O
Molecular Formula
C19H20F3N5O5S2
Molecular Weight
519.52
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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Alternative Products

CatalogName
M11939-01TAK-243
A20369-2TAK-243 2mg
A20369-50TAK-243 50mg
A20369-100TAK-243 100mg
A20369-25TAK-243 25mg
HY-100487RTAK-243 (Standard)
A20369-1TAK-243 1mg
A20369-5TAK-243 5mg
A20369-10TAK-243 10mg
C13356-01TAK-243 (MLN7243)

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