SHU 9119

• Target:

  Others|||Melanocortin Receptor

• Related Pathways:

  Neuroscience|||GPCR/G Protein|||Others

• Bioactivity:

  SHU 9119 is an effective human melanocortin 3 and 4 receptors (MC3/4R) antagonist and a partial MC5R agonist (IC50: 0.23, 0.06, and 0.09 nM for human MC3R, MC4R and MC5R, respectively) .

• Smiles:

  CCCC[C@H](NC(C)=O)C(=O)N[C@H]1CC(=O)NCCCC[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NC(=O)[C@H](Cc2cnc[nH]2)NC1=O)C(N)=O

• Molecular Formula:

  C54H71N15O9

• Molecular Weight:

  1074.258

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  168482-23-3