OSMI-1

• Target:

  Acyltransferase|||Transferase

• Related Pathways:

  Metabolism

• Purity:

  0.9983

• Bioactivity:

  OSMI-1 is an O-GlcNAc transferase (OGT) inhibitor (IC50=2.7 ?M) that is orally active and cell-permeable. OSMI-1 inhibits protein O-GlcNA acetylation without qualitatively altering cell-surface N- or O- linked glycans.

• Smiles:

  COc1ccccc1C(NS(=O)(=O)c1ccc2[nH]c(=O)ccc2c1)C(=O)N(Cc1ccco1)Cc1cccs1

• Molecular Formula:

  C28H25N3O6S2

• Molecular Weight:

  563.64

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1681056-61-0