Products for Research Use Only

Ogerin

CAT: 0931-T16378-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T16378-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1309198-71-7
Target
GPCR, Adenosine Receptor, 5-HT Receptor
Related Pathways
Neuroscience, Endocrinology/Hormones, GPCR/G Protein
Purity
0.999
Bioactivity
Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83) that blocks recall in fear conditioning in mice. It exhibits inverse agonist and antagonist activity (Ki, 220 nM) at the A2A receptor and weak antagonist activity (Ki, 736 nM) at the 5-HT2B receptor.
Smiles
Nc1nc(NCc2ccccc2)nc(n1)-c1ccccc1CO
Molecular Formula
C17H17N5O
Molecular Weight
307.35
Shipping Conditions
Ice Packs
Storage Temperature
-20°C