LP-935509

CAT: 0931-MF-0033199-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0033199-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1454555-29-3
Target
AAK1|||AAK1 (AP2 associated kinase 1) |||Serine/threonin kinase|||SARS-CoV
Related Pathways
Microbiology/Virology|||Metabolism|||Cell Cycle/Checkpoint|||Neuroscience
Purity
0.9964
Bioactivity
LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1) with an IC50 of 3.3 nM and a Ki of 0.9 nM. LP-935509 is a potent inhibitor of BIKE (IC50 of 14 nM) and a moderate inhibitor of GAK (IC50 of 320±40 nM) .
Smiles
COc1ncccc1-c1cnn2ccc(nc12)N1CCN(CC1)C(=O)OC(C)C
Molecular Formula
C20H24N6O3
Molecular Weight
396.44
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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