LP-935509

• Target :

  AAK1|||AAK1 (AP2 associated kinase 1) |||Serine/threonin kinase|||SARS-CoV

• Related Pathways :

  Microbiology/Virology|||Metabolism|||Cell Cycle/Checkpoint|||Neuroscience

• Purity :

  0.9964

• Bioactivity :

  LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1) with an IC50 of 3.3 nM and a Ki of 0.9 nM. LP-935509 is a potent inhibitor of BIKE (IC50 of 14 nM) and a moderate inhibitor of GAK (IC50 of 320±40 nM) .

• Smiles :

  COc1ncccc1-c1cnn2ccc(nc12)N1CCN(CC1)C(=O)OC(C)C

• Molecular Formula :

  C20H24N6O3

• Molecular Weight :

  396.44

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1454555-29-3