RegisterLogin

GSK8814

CAT: 0931-T15443-01Size: 100 mgDry Ice: NoHazardous: No
CAT#:0931-T15443-01Size:100 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
CAS Number
1997369-78-4
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Bioactivity
GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan) . GSK8814 displays 500-fold selectivity for ATAD2 over BRD4 BD1. GSK8814 binds to ATAD2 and BRD4 BD1 (pIC50s: 7.3 and 4.6) .
Smiles
CO[C@H]1CNC[C@@H](OCC2CCC(F)(F)CC2)[C@@H]1Nc1ncc(-c2cncc(C)c2)c2cc(C)c(=O)[nH]c12
Molecular Formula
C28H35F2N5O3
Molecular Weight
527.61
Shipping Conditions
Cool pack
Storage Temperature
-20°C

Related Products

CatalogName
T5540-01GSK8612
T24115-01GSK854
T88845-01GSK484
T32012GSK984
T6852-01GSK481
T15442-01GSK864
T211698-01GSK484-Ph
TQ0067-01GSK484 hydrochloride

Alternative Products

CatalogName
MBS3603118-01GSK8814
A24441-1GSK8814 1mg
A24441-10GSK8814 10mg
A24441-50GSK8814 50mg
A24441-5GSK8814 5mg

Popular Products