GS-626510

CAT: 0931-T15419-01Size: 1 mL - 10 mM (in DMSO)Dry Ice: NoHazardous: No

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CAT#:0931-T15419-01Size:1 mL - 10 mM (in DMSO)

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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CAS Number

1637770-13-8

Target

Epigenetic Reader Domain

Related Pathways

Chromatin/Epigenetic

Bioactivity

GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2) .

Smiles

Cc1noc(C)c1-c1cc(-c2c(C)ccc3ncccc23)c2[nH]c(nc2c1)C1CC1

Molecular Formula

C25H22N4O

Molecular Weight

394.47

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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