GS-626510

• Target:

  Epigenetic Reader Domain

• Related Pathways:

  Chromatin/Epigenetic

• Bioactivity:

  GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2) .

• Smiles:

  Cc1noc (C) c1-c1cc (-c2c (C) ccc3ncccc23) c2[nH]c (nc2c1) C1CC1

• Molecular Formula:

  C25H22N4O

• Molecular Weight:

  394.47

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1637770-13-8