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Apinocaltamide

CAT: 0931-T14120-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0931-T14120-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1838651-58-3
Target
Calcium Channel
Related Pathways
Metabolism, Membrane transporter/Ion channel
Purity
0.998
Bioactivity
Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that penetrates the blood-brain barrier (BBB) with IC50=6.4-18nM for Cav3.1, Cav3.2, and Cav3.3, and is commonly used in epilepsy research.
Smiles
N#CC1=CN=C(C=C1)CN2N=C(C=C2)NC(=O)CC3=CC=C(C=C3)C4(CC4)C(F)(F)F
Molecular Formula
C22H18F3N5O
Molecular Weight
425.41
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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