AP5

• Target :

  Others|||GPCR

• Related Pathways :

  GPCR/G Protein|||Others|||Endocrinology/Hormones

• Bioactivity :

  AP5 is a potent and selective agonist for the GPR40 receptor with positive allosteric modulation of endogenous ligands (AgoPAM) . AP5 demonstrates a rat hIP1 EC50 of 0.49 nM against the GPR40 receptor.

• Smiles :

  [C@@H]([C@@H](C(O)=O)C)(C=1C=C2C(=CC1)CC[C@H](O2)C3=C(F)C=C(C=C3)C=4C=C(OC)N=CC4)[C@H]5CC5

• Molecular Formula :

  C28H28FNO4

• Molecular Weight :

  461.52

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1623194-37-5