Sitaxsentan

• Target :

  Endothelin Receptor

• Related Pathways :

  GPCR/G Protein

• Purity :

  0.9934

• Bioactivity :

  Sitaxsentan (TBC-11251) is A selective endothelin A (ETA) receptor antagonist. Endothelin is an effective vasoconstrictor. Sitaxsentan blocks the binding of endothelin to its receptors, thereby eliminating the harmful effects of endothelin.

• Smiles :

  C(CC=1C=C2C(=CC1C)OCO2)(=O)C3=C(S(NC4=C(Cl)C(C)=NO4)(=O)=O)C=CS3

• Molecular Formula :

  C18H15ClN2O6S2

• Molecular Weight :

  454.9

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  184036-34-8