SGC-iMLLT

• Target :

  Epigenetic Reader Domain|||Histone Methyltransferase

• Related Pathways :

  Chromatin/Epigenetic

• Purity :

  0.9992

• Bioactivity :

  SGC-iMLLT is a potent and selective MLLT1/3-histone interactions inhibitor (IC50 = 0.26 ?M), and is a first-in-class chemical probe displaying cellular target engagement of MLLT1 (Kd = 0.129??M) and MLLT3 (Kd = 0.077??M) .

• Smiles :

  C[C@H]1CCCN1Cc1nc2cc(NC(=O)c3ccc4n(C)ncc4c3)ccc2[nH]1

• Molecular Formula :

  C22H24N6O

• Molecular Weight :

  388.47

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2255338-25-9