PF-06726304
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


PF-06726304
Target:
Histone MethyltransferaseRelated Pathways:
Chromatin/EpigeneticPurity:
0.9954Bioactivity:
PF-06726304 shows robust antitumor growth activity. PF-06726304 is an effective and selective EZH2 inhibitor. PF-06726304 inhibits wild-type and Y641N mutant EZH2 (Kis: 0.7 and 3.0 nM, respectively) .Smiles:
Cc1noc(C)c1-c1cc(Cl)c2CCN(Cc3c(C)cc(C)[nH]c3=O)C(=O)c2c1ClMolecular Formula:
C22H21Cl2N3O3Molecular Weight:
446.33Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
1616287-82-1
