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Alvimopan

CAT: 0931-T1242-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-T1242-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
156053-89-3
Target
Opioid Receptor
Related Pathways
GPCR/G Protein|||Neuroscience|||Endocrinology/Hormones
Purity
0.9997
Bioactivity
Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4- (3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity. Alvimopan is a selective and competitive antagonist at mu-opioid receptors, found in myenteric and submucosal neurons and the immune cells of the lamina propria in the human gut. Upon administration, this agent binds to mu-opioid receptors in the gut, thereby reversing opioid-related disturbances in gut motility. Alvimopan is approximately three to nine times more potent than naloxone.
Smiles
C[C@H]1CN(C[C@H](Cc2ccccc2)C(=O)NCC(O)=O)CC[C@@]1(C)c1cccc(O)c1
Molecular Formula
C25H32N2O4
Molecular Weight
424.53
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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