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GKI-1

CAT: 0931-T11402-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T11402-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2444764-03-6
Target
ROCK, Others
Related Pathways
Stem Cells, Others, Cell Cycle/Checkpoint, Cytoskeletal Signaling
Purity
0.9996
Bioactivity
GKI-1 is a Greatwall (GWL) kinase inhibitor with an IC50 of 4.9 for hGWLFL and 2.5 μM for hGWL-KinDom. It exhibits stronger inhibition on ROCK1 with an IC50 of 11 μM and only weakly inhibits PKA.
Smiles
N(C=1C=C(C=CC1)C=2C=NNC2)C3=CC=C(Cl)C=C3
Molecular Formula
C15H12ClN3
Molecular Weight
269.73
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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Alternative Products

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BUP05214-01GKI-1
BUP11602-01GKI-1 HCl
HY-100521RGKI-1 (Standard)
OF59775-011,1,1,1,1-Kestoheptaose
N2864-5.11,1,1,1-Kestohexaose
1120401,1,1,1-Kestohexose

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