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Giredestrant tartrate

CAT: 0931-T11236-01Size: 500 mgDry Ice: NoHazardous: No
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CAT#:0931-T11236-01Size:500 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2407529-33-1
Target
Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Purity
>99.99%
Bioactivity
Giredestrant tartrate (Estrogen receptor antagonist 1) is a novel, orally active, selective and effective non-steroidal estrogen receptor antagonist. Giredestrant tartrate strongly binds to ER, resulting in the failure of ER to activate the transcription of targeted genes and promoting the degradation of ER protein. Giredestrant tartrate can be used to treat tumor diseases.
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[C@@H]([C@H](C(O)=O)O)(C(O)=O)O.C(C(CO)(F)F)N1[C@@H](C2=C(C=3C(N2)=CC=CC3)C[C@H]1C)C4=C(F)C=C(NC5CN(CCCF)C5)C=C4F
Molecular Formula
C31H37F5N4O7
Molecular Weight
672.64
Shipping Conditions
Ice Packs
Storage Temperature
-20°C