(E) -GABAB receptor antagonist 1

• CAS Number :

  1611483-29-4

• Target :

  GABA Receptor|||ERK

• Related Pathways :

  Membrane transporter/Ion channel|||MAPK|||Neuroscience

• Purity :

  0.9809

• Bioactivity :

  (E) -GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist that decreases GABA-induced IP3 (inositol trisphosphate) production with an IC50 of 37.9 ?M. It is a selective and negative allosteric modulator of GABAB (?-Aminobutyric acid) receptors.

• Smiles :

  C(=C/C(C(O)=O)=O)\C1=CC(C(C)(C)C)=C(O)C(C(C)(C)C)=C1

• Molecular Formula :

  C18H24O4

• Molecular Weight :

  304.38

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C