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Aprocitentan D4

CAT: 0931-T10351-01Size: 100 mgDry Ice: NoHazardous: No
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CAT#:0931-T10351-01Size:100 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Bioactivity
Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM; pA2s: 6.7 and 5.5) .
Smiles
O=S(N)(NC1=NC=NC(OC([2H])([2H])C([2H])([2H])OC2=NC=C(Br)C=N2)=C1C3=CC=C(Br)C=C3)=O
Molecular Formula
C16H10D4Br2N6O4S
Molecular Weight
550.22
Shipping Conditions
Ice Packs
Storage Temperature
-20°C