PPARγ Antagonist, G3335
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PPARγ Antagonist, G3335
Description:
Cell-permeable. A dipeptide that acts as a selective and reversible PPARγ antagonist (KD ~ 8 µM). Shown to inhibit the agonist activity of Rosiglitazone (100 nM) in a dose-dependent manner (IC₅₀ = 31.9 µM) in transfected COS-7 cells.Shipping Conditions:
gel packStorage Conditions:
-20°CShelf Life:
60 months
