PPARγ Antagonist, G3335

CAT:
26-1979-25
Size:
25 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
PPARγ Antagonist, G3335 - image 1

PPARγ Antagonist, G3335

  • Description:

    Cell-permeable. A dipeptide that acts as a selective and reversible PPARγ antagonist (KD ~ 8 µM). Shown to inhibit the agonist activity of Rosiglitazone (100 nM) in a dose-dependent manner (IC₅₀ = 31.9 µM) in transfected COS-7 cells.
  • Shipping Conditions:

    gel pack
  • Storage Conditions:

    -20°C
  • Shelf Life:

    60 months