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VD5123

CAT: 0804-HY-161371Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-161371Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
VD5123 is a serine protease inhibitor. VD5123 inhibits TMPRS2, HGFA, matriptase, hepsin with IC50s of 15, 3980, 140, 37 nM respectively. VD5123 can be used for antiviral research, such as SARS-CoV-2 and broad panel of coronaviruses and influenza viruses[1].
UNSPSC
12352005
Target
Ser/Thr Protease
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/vd5123.html
Solubility
10 mM in DMSO
Smiles
CC(N[C@H](C(N[C@H]1CC(C)C)=O)CC2=CC=C(OC3=CC=CC(C[C@@H](C(N[C@@H](CCCNC(N)=N)C(C4=NC(C=CC=C5)=C5S4)=O)=O)NC1=O)=C3)C=C2)=O
Molecular Formula
C39H46N8O6S
Molecular Weight
754.90
References & Citations
[1]Damalanka VC, et al. Mechanism-Based Macrocyclic Inhibitors of Serine Proteases. J Med Chem. 2024 Mar 13.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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