(+)-MK 801 Hydrogen Maleate
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Catalog number
B2326-5
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Price
Please ask
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Size
5 mg
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Alternative_name
10,11-dihydro-5S-methyl-5H-dibenzo[a,d]cyclohepten-5,10-imine, (2Z)-2-butenedioate,Dizocilpine
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Description
A potent, selective and non-competitive N-methyl-D-aspartate (NMDA) receptor antagonist (Ki = 30.5 nM) that acts at the NMDA receptor-operated ion channel as an open channel blocker, preventing Ca2+ flux. It has been shown to be protective in various models of ischemia as well as to inhibit behavioral sensitization to certain psychostimulants.
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CAS Number
77086-22-7
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Structure Available
Yes
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Molecular Formula
C₂₀H₁₉NO₄
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Molecular Weight
337.37
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Cell Permeable
Yes
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Purity
≥98% by HPLC
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Solubilities
~6 mg/ml (H₂O) in 0,>20 mg/ml (DMSO) in 0
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Handling
Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.
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Tag Line
A potent, selective and non-competitive N-methyl-D-aspartate (NMDA) receptor antagonist
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Storage Condition
-20ºC
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Shipping Condition
Gel Pack
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Shelf Life
36 months
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MDL Number
MFCD0082465
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PubChem CID
6420042
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SMILES
CC12C3=CC=CC=C3CC(N1)C4=CC=CC=C24.C(=CC(=O)O)C(=O)O
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InChi
InChI=1S/C16H15N.C4H4O4/c1-16-13-8-4-2-6-11(13)10-15(17-16)12-7-3-5-9-14(12)16;5-3(6)1-2-4(7)8/h2-9,15,17H,10H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-/t15-,16+;/m1./s1
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InChi Key
QLTXKCWMEZIHBJ-PJGJYSAQSA-N
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MSDS Available
1
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