BRD4770

• Catalog number
  9525-5
• Price
  Please ask
• Size
  5 mg

• Alternative_name
  Methyl 2-benzamido-1-(3-phenylpropyl)-1H-benzo[d]imidazole-5-carboxylate
• Description
  BRD4770 is a selective inhibitor of the histone methyltransferase G9a (also named euchromatin histone methyltransferase 2 (EHMT2). BRD4770 blocks lysine residue 9 methylation of histone H3 without inducing apoptosis. In addition, it induces senescence, and inhibits both anchorage-dependent and -independent proliferation in the pancreatic cancer cell line PANC-1.
• CAS Number
  1374601-40-7
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₂₅H₂₃N₃O₃
• Molecular Weight
  413.47
• Cell Permeable
  Yes
• Purity
  ≥98% by HPLC
• Solubilities
  DMSO(10 mg/ml)
• Handling
  Protect from air and light
• Tag Line
  An inhibitor of histone methyltransferase G9a
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• PubChem CID
  72193870
• PubChem CID Link
• SMILES
  COC(=O)C1=CC2=C(C=C1)N(C(=N2)NC(=O)C3=CC=CC=C3)CCCC4=CC=CC=C4
• InChi
  InChI=1S/C25H23N3O3/c1-31-24(30)20-14-15-22-21(17-20)26-25(27-23(29)19-12-6-3-7-13-19)28(22)16-8-11-18-9-4-2-5-10-18/h2-7,9-10,12-15,17H,8,11,16H2,1H3,(H,26,27,29)
• InChi Key
  UCGWYCMPZXDHNR-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  BRD4770  
• Short name
  BRD4770
• Alternative name
  BRD4770

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