Amlodipine besylate

  • Catalog number
    2378-50
  • Price
    Please ask
  • Size
    50 mg
  • Alternative_name
    2-[(2-Aminoethoxy)methyl]-4-(2-chlo­rophenyl)-1,4-dihydro-6-methyl-3,5-pyridinedicarbo­xylic acid 3-ethyl 5-methyl ester benzenesulfonate
  • Description
    A L-type calcium channel blocker and an anti-hypertensive agent. Amlodipine displays vasoprotective effects in cardiovascular disease and inhibits Ca²⁺-induced contractions in depolarized rat aorta (IC₅₀ = 1.9 nM). Amlodipin also inhibits proliferation of human vascular smooth muscle cells and epidermoid carcinoma A431 cells (IC₅₀ = 25 μM).
  • CAS Number
    111470-99-6
  • Structure Available
    Yes
  • Salt Form
    No
  • Molecular Formula
    C₂₀H₂₅ClN₂O₅.C₆H₆O₃S
  • Molecular Weight
    567.05
  • Cell Permeable
    Yes
  • Purity
    ≥98% by HPLC
  • Solubilities
    DMSO (~100 mM) or H₂O (~10 mM)
  • Handling
    Protect from light and moisture
  • Tag Line
    A calcium channel blocker
  • Storage Condition
    +4°C
  • Shipping Condition
    gel pack
  • Shelf Life
    36 months
  • MDL Number
    MFCD00887594
  • PubChem CID
    60496
  • SMILES
    CCOC(=O)C1=C(NC(=C(C1C2=CC=CC=C2Cl)C(=O)OC)C)COCCN.C1=CC=C(C=C1)S(=O)(=O)O
  • InChi
    InChI=1S/C20H25ClN2O5.C6H6O3S/c1-4-28-20(25)18-15(11-27-10-9-22)23-12(2)16(19(24)26-3)17(18)13-7-5-6-8-14(13)21;7-10(8,9)6-4-2-1-3-5-6/h5-8,17,23H,4,9-11,22H2,1-3H3;1-5H,(H,7,8,9)
  • InChi Key
    ZPBWCRDSRKPIDG-UHFFFAOYSA-N
  • MSDS Available
    Yes
  • Gene target
  • Short name
    Amlodipine besylate
  • Alternative name
    Amlodipine besylate
Product images
Similar products
Filters
Contact
Chat with gentaur.com employee