Y15

• Catalog number
  B1252-50
• Price
  Please ask
• Size
  50 mg

• Alternative_name
  1,2,4,5-benzenetetramine, tetrahydrochloride
• Description
  Y15 is a selective focal adhesion kinase (FAK) inhibitor preventing FAK autophosphorylation at IC₅₀ of 1 μM. It does not have any significant activity against a range of other kinases like EGFR, PDGFR, and IG-RI. Y15 has shown to promote cell detachment inhibiting cell adhesion in in vitro experiments, shows antiproliferative activity in variety of tumor cell lines. In vivo it has shown to inhibit the proliferation in breast cancer cells.
• CAS Number
  4506-66-5
• Structure Available
  Yes
• Salt Form
  Yes
• Molecular Formula
  C₆H₁₀N₄•4HCl
• Molecular Weight
  284.01
• Cell Permeable
  Yes
• Purity
  ≥95%
• Solubilities
  DMSO (>20 mg/ml) or (H₂O (>15 mg/ml)
• Handling
  Protect from air and moisture
• Tag Line
  A selective focal adhesion kinase (FAK) inhibitor having antiproliferative activity
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• MDL Number
  MFCD00012970
• PubChem CID
  78260
• PubChem CID Link
• SMILES
  C1=C(C(=CC(=C1N)N)N)N.Cl.Cl.Cl.Cl
• InChi
  InChI=1S/C6H10N4.4ClH/c7-3-1-4(8)6(10)2-5(3)9;;;;/h1-2H,7-10H2;4*1H
• InChi Key
  BZDGCIJWPWHAOF-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  Y15  
• Short name
  Y15
• Alternative name
  Y15

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