PIK75

• Catalog number
  B1668-25
• Price
  Please ask
• Size
  25 mg

• Alternative_name
  PIK75 , PIK75; PIK 75; PIK-75 Hydrochloride; PIK75 Hydrochloride; PIK 75 Hydrochloride; (E)-N'-((6-bromoH-imidazo[1,2-a]pyridin-3-yl)methylene)-N,2-dimethyl-5-nitrobenzenesulfonohydrazide hydrochloride; PIK-75 Hydrochloride; PIK75 Hydrochloride; PIK 75 Hydrochloride
• Description
  PIK-75 is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM.
• CAS Number
  372196-77-5
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₁₆H₁₅BrClN₅O₄S
• Molecular Weight
  488.74
• Cell Permeable
  Yes
• Purity
  >98%
• Solubilities
  DMSO
• Handling
  Protect from air and light
• Tag Line
  Inhibitor of PI3K isoform p110α
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• MDL Number
  MFCD12546130
• PubChem CID
  45265864
• PubChem CID Link
• SMILES
  CC1=C(C=C(C=C1)[N+](=O)[O-])S(=O)(=O)N(C)N=CC2=CN=C3N2C=C(C=C3)Br.Cl
• InChi
  InChI=1S/C16H14BrN5O4S.ClH/c1-11-3-5-13(22(23)24)7-15(11)27(25,26)20(2)19-9-14-8-18-16-6-4-12(17)10-21(14)16;/h3-10H,1-2H3;1H/b19-9+;
• InChi Key
  VOUDEIAYNKZQKM-MYHMWQFYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  PIK75  
• Short name
  PIK75
• Alternative name
  PIK75

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