GSK180736A
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Catalog numberB1628-5
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PricePlease ask
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Size5 mg
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Alternative_nameGSK180736A; GSK 180736A; GSK-180736A; 4-(4-fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
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DescriptionGSK180736A is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 μM.
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CAS Number817194-38-0
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Structure AvailableYes
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Salt FormNo
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Molecular FormulaC₁₉H₁₆FN₅O₂
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Molecular Weight365.36
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Cell PermeableYes
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Purity>98%
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SolubilitiesDMSO
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HandlingProtect from air and light
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Tag LineA potent and selective inhibitor of GRK2
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Storage Condition-20°C
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Shipping Conditiongel pack
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Shelf Life36 months
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MDL NumberNA
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PubChem CID11233873
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SMILESCC1=C(C(NC(=O)N1)C2=CC=C(C=C2)F)C(=O)NC3=CC4=C(C=C3)NN=C4
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InChi1S/C19H16FN5O2/c1-10-16(17(24-19(27)22-10)11-2-4-13(20)5-3-11)18(26)23-14-6-7-15-12(8-14)9-21-25-15/h2-9,17H,1H3,(H,21,25)(H,23,26)(H2,22,24,27)
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InChi KeyHEAIGWIZTYAQTC-UHFFFAOYSA-N
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MSDS AvailableYes
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Gene target
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Short nameGSK180736A
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Alternative nameGSK180736A
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