XMD17-109

• Catalog number
  B1685-5
• Price
  Please ask
• Size
  5 mg

• Alternative_name
  XMD17-109; XMD17 109; XMD17109; 11-cyclopentyl-2-[2-ethoxy-4-[4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]anilino]-5-methylpyrimido[4,5-b][1,4]benzodiazepin-6-one
• Description
  XMD17-109 is a novel, specific ERK-5 inhibitor, which inhibits the ERK5-mediated AP1 transcriptional activity at 30 μM, and has an EC50 of 4.2 μM.
• CAS Number
  1435488-37-1
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₃₆H₄₆N₈O₃
• Molecular Weight
  638.8
• Cell Permeable
  Yes
• Purity
  >98%
• Solubilities
  DMSO
• Handling
  Protect from air and light
• Tag Line
  A ERK-5 inhibitor
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• MDL Number
  NA
• PubChem CID
  71604307
• PubChem CID Link
• SMILES
  CCOC1=C(C=CC(=C1)C(=O)N2CCC(CC2)N3CCN(CC3)C)NC4=NC=C5C(=N4)N(C6=CC=CC=C6C(=O)N5C)C7CCCC7
• InChi
  InChI=1S/C36H46N8O3/c1-4-47-32-23-25(34(45)43-17-15-26(16-18-43)42-21-19-40(2)20-22-42)13-14-29(32)38-36-37-24-31-33(39-36)44(27-9-5-6-10-27)30-12-8-7-11-28(30)35(46)41(31)3/h7-8,11-14,23-24,26-27H,4-6,9-10,15-22H2,1-3H3,(H,37,38,39)
• InChi Key
  XVBGRTMNFNMINE-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  XMD17-109  
• Gene symbol
  TMED7, OR7E110P
• Short name
  XMD17-109
• Alternative name
  XMD17-109

Gene info

• Identity
  HGNC:24253
• Gene
  TMED7
• Long gene name
  transmembrane p24 trafficking protein 7
• Synonyms gene name
  • transmembrane emp24 protein transport domain containing 7
• Synonyms
  • CGI-109
  • FLJ90481
  • p24gamma3
  • p24g3
• GenBank acession
  • AK074962
• Locus
  5q22.3
• Discovery year
  2004-12-21
• Entrez gene record
  51014
• Pubmed identfication
  • 10810093
• RefSeq identity
  • NM_181836
• Classification
  • Transmembrane p24 trafficking proteins
• VEGA ID
  OTTHUMG00000132013

Gene info

• Identity
  HGNC:15126
• Gene
  OR7E110P
• Long gene name
  olfactory receptor family 7 subfamily E member 110 pseudogene
• Synonyms gene
  • OR7E68P
  • OR7E71P
  • OR7E72P
  • OR7E73P
  • OR7E74P
  • OR7E75P
• Synonyms gene name
  • olfactory receptor, family 7, subfamily E, member 110 pseudogene
• Synonyms
  • hg674
  • OR912-109
  • OR912-46
  • OR912-108
  • OR912-110
  • hg523
• Locus
  10p13
• Discovery year
  2001-03-28
• Entrez gene record
  81354
• Classification
  • Olfactory receptors, family 7
• VEGA ID
  OTTHUMG00000017715

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