GSK-3787

• Catalog number
  2400-25
• Price
  Please ask
• Size
  25 mg

• Alternative_name
  4-Chloro-N-(2-{[5-(trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide
• Description
  GSK-3787 is a selective and irreversible antagonist of the peroxisome proliferator-activated receptor delta (PPARδ) (plC₅₀ = 6.6). It covalently binds to Cys 249 in the PPARδ binding site.
• CAS Number
  188591-46-0
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₁₅H₁₂ClF₃N₂O₃S
• Molecular Weight
  392.78
• Cell Permeable
  Yes
• Purity
  ≥98% by TLC
• Solubilities
  DMSO (~30 mg/ml)
• Handling
  Protect from light and air
• Tag Line
  A potent PPARδ antagonist
• Storage Condition
  -20 ̊C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• MDL Number
  MFCD00099612
• PubChem CID
  2800647
• PubChem CID Link
• SMILES
  C1=CC(=CC=C1C(=O)NCCS(=O)(=O)C2=NC=C(C=C2)C(F)(F)F)Cl
• InChi
  InChI=1S/C15H12ClF3N2O3S/c16-12-4-1-10(2-5-12)14(22)20-7-8-25(23,24)13-6-3-11(9-21-13)15(17,18)19/h1-6,9H,7-8H2,(H,20,22)
• InChi Key
  JFUIMTGOQCQTPF-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  GSK-3787  
• Short name
  GSK-3787
• Alternative name
  GSK-3787

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