PF-04981517

• Catalog number
  2917-5
• Price
  Please ask
• Size
  5 mg

• Alternative_name
  1-methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-(1-piperidinyl)-1-pyrrolidinyl]-1H-pyrazolo[3,4-d]pyrimidine, CYP3cide
• Description
  Potent and selective inhibitor of CYP3A (IC50 = 30 nM (CYP3A4), 17 μM (CYP3A5) and 70 μM (CYP3A7).
• CAS Number
  1390637-82-7
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₂₆H₃₂N₈
• Molecular Weight
  456.6
• Cell Permeable
  Yes
• Purity
  ≥98%
• Solubilities
  DMSO (~20 mg/ml), DMF (~30 mg/ml), Ethanol (~2 mg/ml)
• Handling
  Protect from air, light and moisture
• Tag Line
  A potent and specific inhibitor of Cytochrome P450 3A
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  24 months
• PubChem CID
  71315139
• PubChem CID Link
• SMILES
  CC1=CC=C(C=C1)C2=C(C=NN2C)C3=NN(C4=C3C(=NC=N4)N5CCC(C5)N6CCCCC6)C
• InChi
  InChI=1S/C26H32N8/c1-18-7-9-19(10-8-18)24-21(15-29-31(24)2)23-22-25(32(3)30-23)27-17-28-26(22)34-14-11-20(16-34)33-12-5-4-6-13-33/h7-10,15,17,20H,4-6,11-14,16H2,1-3H3/t20-/m0/s1
• InChi Key
  WDWIMDKOXZZYHH-FQEVSTJZSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  PF-04981517  
• Short name
  PF-04981517
• Alternative name
  PF-04981517

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