Lasofoxifene tartrate
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Catalog number9680-5
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PricePlease ask
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Size5 mg
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Alternative_name(5R,6S)-5,6,7,8-tetrahydro-6-phenyl-5-[4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-2-naphthalenol, (2S,3S)-2,3-dihydroxybutanedioate; CP-336,156
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DescriptionLasofoxifene is a unique, non-steroidal selective estrogen receptor modulator (SERM). It selectively binds to human ERα with an IC₅₀ value of 1.5 nM and inhibits bone loss in ovariectomized rats. Has potential use in treating breast cancer.
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CAS Number190791-29-8
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Structure AvailableYes
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Salt FormNo
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Molecular FormulaC₂₈H₃₁NO₂.C₄H₆O₆
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Molecular Weight563.6
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Cell PermeableYes
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Purity≥98% by HPLC
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SolubilitiesDMSO (>5 mg/ml)
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HandlingProtect from air and moisture
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Tag LineA non-steroidal selective estrogen receptor modulator (SERM)
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Storage Condition-20°C
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Shipping Conditiongel pack
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Shelf Life36 months
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PubChem CID3081919
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SMILESC1CCN(C1)CCOC2=CC=C(C=C2)C3C(CCC4=C3C=CC(=C4)O)C5=CC=CC=C5.C(C(C(=O)O)O)(C(=O)O)O
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InChiInChI=1S/C28H31NO2.C4H6O6/c30-24-11-15-27-23(20-24)10-14-26(21-6-2-1-3-7-21)28(27)22-8-12-25(13-9-22)31-19-18-29-16-4-5-17-29;5-1(3(7)8)2(6)4(9)10/h1-3,6-9,11-13,15,20,26,28,30H,4-5,10,14,16-19H2;1-2,5-6H,(H,7,8)(H,9,10)/t26-,28+;1-,2-/m10/s1
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InChi KeyINEHJXCWEVNEDZ-LUDNRVPPSA-N
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MSDS AvailableYes
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Gene target
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Short nameLasofoxifene tartrate
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Alternative nameLasofoxifene tartrate
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