PIK-294

• Catalog number
  2614-5
• Price
  Please ask
• Size
  5 mg

• Alternative_name
  2-[[4-Amino-3-(3-hydroxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]methyl]-5-methyl-3-(2-methylphenyl)-4(3H)-quinazolinone
• Description
  PIK-294 is a highly potent and selective p110δ inhibitor (IC₅₀ of 10 nM). Displays 1000-, 49- and 16-fold less potency against PI3Kα/β/γ, respectively.
• CAS Number
  900185-02-6
• Structure Available
  Y
• Salt Form
  No
• Molecular Formula
  C₂₈H₂₃N₇O₂
• Molecular Weight
  489.53
• Cell Permeable
  Yes
• Purity
  >98% by HPLC
• Solubilities
  DMSO (>60 mg/ml)
• Handling
  Protect from air and light
• Tag Line
  A potent PI3K p110δ inhibitor
• Storage Condition
  -20 ̊C
• Shipping Condition
  Gel pack
• Shelf Life
  36 months
• PubChem CID
  24905149
• PubChem CID Link
• SMILES
  O=C1N(C2=CC=CC=C2C)C(CN3N=C(C4=CC=CC(O)=C4)C5=C(N)N=CN=C53)=NC6=C1C(C)=CC=C6
• InChi
  InChI=1S/C28H23N7O2/c1-16-7-3-4-12-21(16)35-22(32-20-11-5-8-17(2)23(20)28(35)37)14-34-27-24(26(29)30-15-31-27)25(33-34)18-9-6-10-19(36)13-18/h3-13,15,36H,14H2,1-2H3,(H2,29,30,31)
• InChi Key
  WFSLJOPRIJSOJR-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  PIK-294  
• Short name
  PIK-294
• Alternative name
  PIK-294

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