Ertugliflozin
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Catalog numberB1896-5
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PricePlease ask
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Size5 mg
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Alternative_name(1S,2S,3S,4R,5S)-5-(4-Chloro-3-(4-ethoxybenzyl)phenyl)-1-hydroxymethyl-6,8-dioxabicyclo(3.2.1)octane-2,3,4-triol; PF-04971729
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DescriptionErtugliflozin is a potent and selective inhibitor of the sodium-dependent glucose cotransporter 2(SGLT2); increases the excretion of glucose with a 2,000-fold selectivity over SGLT1 (IC₅₀ = 0.877 and 1,960 nM, respectively, for human isoforms in vitro.
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CAS Number1210344-57-2
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Structure AvailableYes
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Salt FormNo
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Molecular FormulaC₂₂H₂₅ClO₇
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Molecular Weight436.89
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Cell PermeableYes
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Purity≥98% by HPLC
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SolubilitiesDMSO
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HandlingProtect from air and light
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Tag LineA potent and selective sodium-dependent glucose cotransporter 2(SGLT2) inhibitor
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Storage Condition-20°C
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Shipping Conditiongel pack
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Shelf Life36 months
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PubChem CID44814423
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SMILESCCOC1=CC=C(C=C1)CC2=C(C=CC(=C2)C34C(C(C(C(O3)(CO4)CO)O)O)O)Cl
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InChiInChI=1S/C22H25ClO7/c1-2-28-16-6-3-13(4-7-16)9-14-10-15(5-8-17(14)23)22-20(27)18(25)19(26)21(11-24,30-22)12-29-22/h3-8,10,18-20,24-27H,2,9,11-12H2,1H3/t18-,19-,20+,21-,22-/m0/s1
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InChi KeyMCIACXAZCBVDEE-CUUWFGFTSA-N
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MSDS AvailableYes
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Gene target
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Short nameErtugliflozin
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Alternative nameErtugliflozin
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