BAG 956

• Catalog number
  2456-25
• Price
  Please ask
• Size
  25 mg

• Alternative_name
  α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyr​idinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-be​nzeneacetonitrile
• Description
  A potent, ATP-competitive, dual PI3K/PDK-1 inhibitor in vitro and in vivo (IC₅₀ = 56, 444, 34, 117 and 240 nM for PI3K p110-α ,β,d, γ, and PDK1 kinases, respectively). Displays anticancer properties.
• CAS Number
  853910-02-8
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₂₈H₂₁N₅
• Molecular Weight
  427.5
• Cell Permeable
  Yes
• Purity
  ≥98% by HPLC
• Solubilities
  DMSO (~15 mg/ml) or EtOH (~7 mg/ml)
• Handling
  Protect from air and light
• Tag Line
  A dual PI3K/PDK-1 inhibitor
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  24 months
• PubChem CID
  24882589
• PubChem CID Link
• SMILES
  CC1=NC2=CN=C3C=CC(=CC3=C2N1C4=CC=C(C=C4)C(C)(C)C#N)C#CC5=CN=CC=C5
• InChi
  InChI=1S/C28H21N5/c1-19-32-26-17-31-25-13-8-20(6-7-21-5-4-14-30-16-21)15-24(25)27(26)33(19)23-11-9-22(10-12-23)28(2,3)18-29/h4-5,8-17H,1-3H3
• InChi Key
  GVPAGJWVBUZHNQ-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  BAG   956  
• Short name
  BAG 956
• Alternative name
  BAG 956

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