MS436
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Catalog number2680-5
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PricePlease ask
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Size5 mg
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Alternative_name(E)-4-[2-(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-N-2-pyridinylbenzenesulfonamide
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DescriptionMS436 is a potent and selective BRD4 bromodomain inhibitor (Ki = 30-50 nM for BrD1). It displays 10-fold selectivity for BrD1 of BRD4 over BrD2 of BRD4.
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CAS Number1395084-25-9
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Structure AvailableY
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Salt FormNo
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Molecular FormulaC₁₈H₁₇N₅O₃S
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Molecular Weight383.42
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Cell PermeableYes
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Purity≥98% by HPLC
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SolubilitiesDMSO (>30 mg/ml)
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HandlingProtect from air and light
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Tag LineA potent BRD4 bromodomain inhibitor
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Storage Condition-20°C
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Shipping ConditionGel pack
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Shelf Life36 months
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PubChem CID60171585
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SMILESCC1=CC(=NNC2=CC=C(C=C2)S(=O)(=O)NC3=CC=CC=N3)C(=CC1=O)N
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InChinChI=1S/C18H17N5O3S/c1-12-10-16(15(19)11-17(12)24)22-21-13-5-7-14(8-6-13)27(25,26)23-18-4-2-3-9-20-18/h2-11,21H,19H2,1H3,(H,20,23)/b22-16-
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InChi KeyBBJDRANVVNBXAR-JWGURIENSA-N
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MSDS AvailableYes
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Gene target
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Short nameMS436
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Alternative nameMS436
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