KT5720
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Catalog number2276-50
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PricePlease ask
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Size50 ug
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Alternative_name(9R,10S,12S)-2,3,9,10,11,12-Hexahydro-10-hydroxy-9-methyl-1-oxo-9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid, hexyl ester
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DescriptionA derivative of the protein kinase inhibitor K252a (Cat. No. 2013). Acts as a potent, selective, ATP-competitive inhibitor of protein kinase A (PKA) (Ki = 60 nM). Has no effect on PKC, PKG and MLCK.
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CAS Number108068-98-0
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Structure AvailableYes
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Salt FormNo
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Molecular FormulaC₃₂H₃₁N₃O₅
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Molecular Weight537.61
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Cell PermeableYes
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Purity≥98% by HPLC
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SolubilitiesDMSO (~50 mM)
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HandlingProtect from air and moisture
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Tag LineA potent and selective Protein kinase A (PKA) inhibitor
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Storage Condition-20 ̊C
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Shipping Conditiongel pack
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Shelf Life24 months
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MDL NumberMFCD00132118
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PubChem CID3844
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SMILESCCCCCCOC(=O)C1(CC2N3C4=CC=CC=C4C5=C6C(=C7C8=CC=CC=C8N(C7=C53)C1(O2)C)CNC6=O)O
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InChiInChI=1S/C32H31N3O5/c1-3-4-5-10-15-39-30(37)32(38)16-23-34-21-13-8-6-11-18(21)25-26-20(17-33-29(26)36)24-19-12-7-9-14-22(19)35(28(24)27(25)34)31(32,2)40-23/h6-9,11-14,23,38H,3-5,10,15-17H2,1-2H3,(H,33,36)
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InChi KeyZHEHVZXPFVXKEY-UHFFFAOYSA-N
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MSDS AvailableYes
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Gene target
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Short nameKT5720
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Alternative nameKT5720
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