GLP-1R agonist 21
CAT:
804-HY-162436
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

GLP-1R agonist 21
- UNSPSC Description: GLP-1R agonist 21 (Compound I-134) is an agonist for glucagon-like peptide-1 receptor (GLP-1 receptor), with EC50 of 0.0104 nM[1].
- Target Antigen: GLP Receptor
- Type: Reference compound
- Related Pathways: GPCR/G Protein
- Applications: Metabolism-protein/nucleotide metabolism
- Field of Research: Metabolic Disease
- Assay Protocol: https://www.medchemexpress.com/glp-1r-agonist-21.html
- Solubility: 10 mM in DMSO
- Smiles: ClC1=CC(F)=C(COC2=C(C(F)F)C=C(CCN(CC3=NC4=C(OC)C=C(C(O)=O)C=C4N3C[C@@H]5CCO5)[C@H]6C)C6=N2)C(F)=C1
- Molecular Weight: 649.03
- References & Citations: [1]Kitamura FY, et al., Fused ring compound having glp-1 receptor agonist effect. WO2024063143A1.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported