CXCR7 modulator 1

CXCR7 modulator 1

• CAS Number: 2231812-31-8
• UNSPSC Description: CXCR7 modulator 1 (compound 25) is a potent and orally bioavailable peptoid hybrid CXCR7 modulator, with a Ki of 9 nM[1].
• Target Antigen: CXCR
• Type: Reference compound
• Related Pathways: GPCR/G Protein;Immunology/Inflammation
• Applications: Metabolism-protein/nucleotide metabolism
• Field of Research: Endocrinology
• Assay Protocol: https://www.medchemexpress.com/cxcr7-modulator-1.html
• Purity: 99.50
• Solubility: DMSO : 250 mg/mL (ultrasonic)
• Smiles: O=C(N[C@@H](CC(C)(C)C)C(N[C@@H](CC1=CSC=N1)C(N2CCC[C@@H]2C(N(CCCC3=C(F)C=C(F)C=C3)CC4=O)=O)=O)=O)[C@@H](CC5=CC=CC=C5)NC([C@H](COCC6=CC=CC=C6)N4)=O
• Molecular Weight: 914.07
• References & Citations: [1]Boehm M, et al. Discovery of Potent and Orally Bioavailable Macrocyclic Peptide-Peptoid Hybrid CXCR7 Modulators. J Med Chem. 2017 Dec 14;60(23):9653-9663.
• Shipping Conditions: Blue Ice
• Storage Conditions: -20°C (Powder, stored under nitrogen)
• Clinical Information: No Development Reported