NPFF2-R ligand 1

• UNSPSC Description:

  NPFF2-R ligand 1 (Compound 16a) is a NPFF2-R ligand, with Kis of 228 and 27 nM for NPFF1-R and NPFF2-R respectively. NPFF2-R ligand 1 can be used for research related with central nervous system[1].

• Target Antigen:

  Others

• Type:

  Reference compound

• Related Pathways:

  Others

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/npff2-r-ligand-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(CCN1CCCCC1)NCC2(CCN(CC3=CC=CC=C3)CC2)CC4=CC=CC5=C4C=CC=C5

• Molecular Weight:

  483.69

• References & Citations:

  [1]Galal KA, et al. Guanidine-to-piperidine switch affords high affinity small molecule NPFF ligands with preference for NPFF1-R and NPFF2-R subtypes. Eur J Med Chem. 2024 Mar 23;269:116330.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported