CPI-169

• Description:

  CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  528.66

• Molecular Formula:

  C27H36N4O5S

• Notes:

  Research use only, not for human use.

• Receptor:

  EZH1| EZH2 WT| EZH2 Y641N

• CAS Number:

  1450655-76-1