PP242

• Catalog number
  1658-1
• Price
  Please ask
• Size
  1 mg

• Alternative_name
  2-(4-Amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-1H-indol-5-ol
• Description
  A potent and selective in vitro mTOR inhibitor that targets the ATP domain of mTOR (IC₅₀ = 8 nM). Inhibits other PI 3-Kinases only at much higher concentrations. Recently it has been shown that PP242 is a more effective mTORC1 inhibitor than Rapamycin (Cat. No. 1568-5 & 1568-50).
• CAS Number
  1092351-67-1
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₁₆H₁₆N₆O
• Molecular Weight
  308.34
• Cell Permeable
  Yes
• Purity
  ≥98% by HPLC
• Solubilities
  DMSO (>50 mg/ml)
• Handling
  Protect from air and light
• Tag Line
  A mTOR inhibitor
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  24 months
• MDL Number
  MFCD12196869
• PubChem CID
  25243800
• PubChem CID Link
• SMILES
  CC(C)N1C2=C(C(=C3C=C4C=C(C=CC4=N3)O)N1)C(=NC=N2)N
• InChi
  InChI=1S/C16H16N6O/c1-8(2)22-16-13(15(17)18-7-19-16)14(21-22)12-6-9-5-10(23)3-4-11(9)20-12/h3-8,21,23H,1-2H3,(H2,17,18,19)/b14-12+
• InChi Key
  MTICIDWIKCANDD-WYMLVPIESA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  PP242  
• Short name
  PP242
• Alternative name
  PP242

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