EPZ011989 for cell activation

EPZ011989 for cell activation is available 2 times from Biovision labs

B1221-25 | EPZ011989 for cell activationsize: 25 mg | 877.21 USD

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B1221-5 | EPZ011989 for cell activationsize: 5 mg | 265.37 USD

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  • Description
    EPZ011989 is a potent EZH2 inhibitor with Ki values that are less than 3 nM for wild type and Tyr646 mutated EZH2. It displays 15-fold selectivity for EZH2 over EZH1 and is without effect against an array of other lysine methyltransferases. EPZ011989 demonstrates significant tumor growth inhibition in a mouse xenograft model of human B cell lymphoma.
  • Peptide sequence
    N/A
  • CAS number
    1598383-40-4
  • Molecular weight
    605.82
  • Category
    Biochemicals
  • Other name
    N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-(ethyl((1r,4r)-4-((2-methoxyethyl)(methyl)amino)cyclohexyl)amino)-2-methyl-5-(3-morpholinoprop-1-yn-1-yl)benzamide
  • Molecular formula
    C₃₅H₅₁N₅O₄ 
  • Physical appearance
    Off-white solid
  • Supplied with
    N/A
  • Is this a salt?
    No
  • Is it cell-permeable?
    Yes
  • Purification
    ≥98% by HPLC
  • Reconstitute instructions
    DMSO(>10 mg/ml)
  • Storage condition
    -20°C
  • Shipping condition
    gel pack
  • Maximum time for storage
    36 months
  • Storage instructions
    Protect from air and light
  • Additional description
    For cells, cell lines and tissues in culture till half confluency.
  • Gene target
  • Short name
    EPZ011989 for activation
  • Technique
    activation
  • Alternative name
    EPZ011989 to measure cellular activation
  • Tissue
    cell
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