DiscoveryPak™ EGFR Tyrosine Kinase Inhibitor Set
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Catalog number
K858-5
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Price
Please ask
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Size
5 inhibitors
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Alternative_name
EGFR Tyrosine Kinase Inhibitor Set, DiscoveryPak™
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Description
A convenient set consisting of five Epidermal Growth Factor Receptor (EGFR) Tyrosine Kinase (TK) inhibitors. The five inhibitors are: 5 mg of Canertinib (Cat. No. 1617-5), 100 mg of Erlotinib, Hydrochloride (Cat. No. 1588-100), 5 mg of Gefitinib (Cat. No. 1589-5), 25 mg of Lapatinib, Ditosylate (Cat. No. 1624-25), and 2 mg of PD 153035 Hydrochloride (Cat. No. 1656-2).
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CAS Number
See under the individual product
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Structure Available
See under the individual product
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Salt Form
No
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Molecular Formula
See under the individual product
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Molecular Weight
See under the individual product
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Cell Permeable
Yes
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Purity
≥95% by HPLC
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Solubilities
DMSO
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Handling
Protect from air, light and moisture
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Tag Line
An EGFR kinase inhibitors set
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Storage Condition
-20°C
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Shipping Condition
gel pack
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Shelf Life
24 months
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SMILES
N/A
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InChi
N/A
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InChi Key
N/A
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MSDS Available
Yes
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Additional description
Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.
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Gene target
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Gene symbol
EGFR-AS1, EGILA, EGFR, RHBDF1
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Short name
DiscoveryPak™ EGFR Tyrosine Kinase Inhibitor Set
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Alternative name
DiscoveryPak™ epidermal growth factor receptor Tyrosine phosphorylation catalyst suppressor Set
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Alternative to gene target
epidermal growth factor receptor, ERBB and ERBB1 and HER1 and mENA and PIG61, EGFR and IDBG-16933 and ENSG00000146648 and 1956, transferase activity, nuclei, Egfr and IDBG-151194 and ENSMUSG00000020122 and 13649, EGFR and IDBG-644035 and ENSBTAG00000011628 and 407217
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Tissue
set
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Gene info
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Identity
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Gene
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Long gene name
EGFR antisense RNA 1
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Locus
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Discovery year
2012-11-06
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Entrez gene record
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Pubmed identfication
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RefSeq identity
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Classification
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VEGA ID
Gene info
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Identity
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Gene
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Long gene name
EGFR interacting lncRNA
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Synonyms
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Locus
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Discovery year
2019-09-27
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Pubmed identfication
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Classification
- Long non-coding RNAs with non-systematic symbols
Gene info
Gene info
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Identity
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Gene
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Long gene name
rhomboid 5 homolog 1
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Synonyms gene
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Synonyms gene name
- chromosome 16 open reading frame 8
- rhomboid family 1 (Drosophila)
- rhomboid 5 homolog 1 (Drosophila)
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Synonyms
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GenBank acession
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Locus
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Discovery year
2003-04-07
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Entrez gene record
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Pubmed identfication
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RefSeq identity
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Classification
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VEGA ID
MeSH Data
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Name
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Concept
Scope note:
A membrane or barrier with micrometer sized pores used for separation purification processes.
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Tree numbers
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Qualifiers
parasitology, microbiology, ethics, virology, trends, veterinary, history, classification, economics, standards, supply & distribution, adverse effects, statistics & numerical data
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