MS023
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Catalog numberB2575-25
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PricePlease ask
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Size25 mg
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Alternative_nameN1-((4-(4-isopropoxyphenyl)-1H-pyrrol-3-yl)methyl)-N1-methylethane-1,2-diamine, MS-023
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DescriptionMS023 is a potent, selective, and cell-active inhibitor of human type I protein arginine methyltransferases (PRMTs) (IC₅₀s of 30, 119, 83, 4 and 5 nM for PRMT1, PRMT3, PRMT4, PRMT6, and PRMT8, respectively). MS023 is completely inactive against type II and type III PRMTs, protein lysine methyltransferases and DNA methyltransferases.
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CAS Number1831110-54-3
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Structure AvailableYes
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Salt FormNo
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Molecular FormulaC₁₇H₂₅N₃O
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Molecular Weight287.41
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Cell PermeableTrue
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Purity≥98% by HPLC
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Solubilities>25 mg/ml in DMSO
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HandlingDo not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.
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Tag LineType I Protein Arginine Methyltransferases inhibitor
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Storage Condition-20ºC
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Shipping ConditionGel Pack
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Shelf Life36 months
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PubChem CID92136227
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SMILESCC(C)OC1=CC=C(C=C1)C2=CNC=C2CN(C)CCN
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InChiInChI=1S/C17H25N3O/c1-13(2)21-16-6-4-14(5-7-16)17-11-19-10-15(17)12-20(3)9-8-18/h4-7,10-11,13,19H,8-9,12,18H2,1-3H3
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InChi KeyFMTVWAGUJRUAKE-UHFFFAOYSA-N
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MSDS AvailableTrue
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Gene target
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Short nameMS023
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Alternative nameMS023
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